201038-58-6
201038-58-6
Chemical Structure
SB 258741
- CAS No.: 201038-58-6
- Formula:C19H30N2O2S
- Molecular Weight:350.52
IUPAC Name: (R)-4-methyl-1-(2-(1-(m-tolylsulfonyl)pyrrolidin-2-yl)ethyl)piperidine
InChIKey: YVWGGGGMRDLOGA-GOSISDBHSA-N
SMILES: O=S(N1[C@@H](CCN2CCC(C)CC2)CCC1)(C3=CC=CC(C)=C3)=O
Biological Activity:
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SB 258741 | SB 258741 is an efficient and highly selective 5-HT7 receptor (pKi = 8. | |||||||||||||||||||||
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References
- Pouzet B, et al. Effects of the 5-HT(7) receptor antagonist SB-258741 in animal models for schizophrenia. Pharmacol Biochem Behav. 2002 Apr;71(4):655-65. [Content Brief]
- Mahé C, et al. Differential inverse agonist efficacies of SB-258719, SB-258741 and SB-269970 at human recombinant serotonin 5-HT7 receptors. Eur J Pharmacol. 2004 Jul 14;495(2-3):97-102. [Content Brief]
Keywords
