2160582-57-8
2160582-57-8
Chemical Structure
Obafistat
- CAS No.: 2160582-57-8
- Formula:C15H16FN5O3S
- Molecular Weight:365.38
IUPAC Name: (8-((3-fluorophenyl)sulfonyl)-3,8-diazabicyclo[3.2.1]octan-3-yl)(1H-1,2,3-triazol-5-yl)methanone
InChIKey: MQFQQVWKRIYYPY-UHFFFAOYSA-N
SMILES: O=C(N1CC(N2S(=O)(C3=CC=CC(F)=C3)=O)CCC2C1)C4=CN=NN4
Biological Activity: Obafistat is a potent aldo-keto reductase AKR1C3 inhibitor with an IC50 of 1.2 nM for human AKR1C3 (patent WO2017202817A1, example 4)[1].
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Obafistat | 99.92% | Obafistat is a potent aldo-keto reductase AKR1C3 inhibitor with an IC50 of 1.2 nM for human AKR1C3 (patent WO2017202817A1, example 4). | ||||||||||||||||||||
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Obafistat (Standard) | ≥98% | Obafistat (Standard) is the analytical standard of Obafistat (HY-109154). This product is intended for research and analytical applications. Obafistat is a potent aldo-keto reductase AKR1C3 inhibitor with an IC50 of 1.2 nM for human AKR1C3 (patent WO2017202817A1, example 4). | ||||||||||||||||||||
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References
Keywords
