2323525-19-3
2323525-19-3
Chemical Structure
uPSEM792
- CAS No.: 2323525-19-3
- Formula:C14H15N3O
- Molecular Weight:241.29
InChIKey: UEUFVUIOCKHRTA-UHFFFAOYSA-N
SMILES: CN1C2=C(C=C(C3CNCC4C3)C4=C2)N=CC1=O
Biological Activity: uPSEM792 is a pharmacologically selective effector molecules (PSEM) agonist for PSAM4-GlyR, with an affinity of Ki of 0.7 nM. uPSEM792 is a substrate for efflux transporters in brains of wild type and dual P-gp and BCRP knockout mice. uPSEM7952 is a possible lead for developing the PET radioligand for PSAM4-GlyR[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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uPSEM792 | 98.02% | uPSEM792 is a pharmacologically selective effector molecules (PSEM) agonist for PSAM4-GlyR, with an affinity of Ki of 0.7 nM. uPSEM792 is a substrate for efflux transporters in brains of wild type and dual P-gp and BCRP knockout mice. uPSEM7952 is a possible lead for developing the PET radioligand for PSAM4-GlyR. | ||||||||||||||||||||
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References
Keywords
