2531244-56-9
Chemical Structure
BJJF078
- CAS No.: 2531244-56-9
- Formula:C27H29N3O6S
- Molecular Weight:523.60
IUPAC Name: N-(5-((4-acrylamidopiperidin-1-yl)sulfonyl)naphthalen-1-yl)-3,4-dimethoxybenzamide
InChIKey: IJRQXDUGUAWTNT-UHFFFAOYSA-N
SMILES: O=C(NC1CCN(S(=O)(C2=C3C=CC=C(NC(C4=CC=C(C(OC)=C4)OC)=O)C3=CC=C2)=O)CC1)C=C
Biological Activity: BJJF078 is an aminopiperidine derivative. BJJF078 is a potent inhibitor of recombinant human and mouse Transglutaminase enzyme (TG2) activity, IC50 values of 41 and 54 nM, respectively. BJJF078 also inhibits the close related enzyme TG1, with an IC50 of 0.16 μM. BJJF078 can be used for Multiple sclerosis (MS) research[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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BJJF078 | 99.66% | BJJF078 is an aminopiperidine derivative. BJJF078 is a potent inhibitor of recombinant human and mouse Transglutaminase enzyme (TG2) activity, IC50 values of 41 and 54 nM, respectively. BJJF078 also inhibits the close related enzyme TG1, with an IC50 of 0.16 μM. BJJF078 can be used for Multiple sclerosis (MS) research. | ||||||||||||||||||||
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Keywords
