2654743-22-1
2654743-22-1
Chemical Structure
MRTX0902
- CAS No.: 2654743-22-1
- Formula:C22H24N6O
- Molecular Weight:388.47
IUPAC Name: 2,5-dihexyl-3,6-bis(5''-hexyl-[2,2':5',2''-terthiophen]-5-yl)-2,5-dihydropyrrolo[3,4-c]pyrrole-1,4-dione
InChIKey: ILPWEAHQRAWJIU-OAHLLOKOSA-N
SMILES: C[C@H](C1=C(C(C#N)=CC=C1)C)NC2=NN=C(C)C3=C2C=C(N4CCOCC4)N=C3
Biological Activity: MRTX0902 is a potent, selective, brain-penetrant, and orally active SOS1 inhibitor with a Ki of 1.9 nM. MRTX0902 disrupts the SOS1:KRASG12C protein-protein interaction (PPI). MRTX0902 can be used in research on pancreatic ductal adenocarcinoma[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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MRTX0902 | 99.67% | MRTX0902 is a potent, selective, brain-penetrant, and orally active SOS1 inhibitor with a Ki of 1.9 nM. MRTX0902 disrupts the SOS1:KRASG12C protein-protein interaction (PPI). MRTX0902 can be used in research on pancreatic ductal adenocarcinoma. | ||||||||||||||||||||
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References
Keywords
