2718990-76-0
2718990-76-0
Chemical Structure
5-HT2A/5-HT2C inverse agonist 1
- CAS No.: 2718990-76-0
- Formula:C24H35N5O2
- Molecular Weight:425.57
InChIKey: HOVLTWZHAUDSGN-QFIPXVFZSA-N
SMILES: CN(C=C1)N=C1CN([C@@H]2C3(CN(CC2)C)CC3)C(NCC4=CC=C(C=C4)OCCC)=O
Biological Activity: 5-HT2A/5-HT2C inverse agonist 1 is a potent and dual 5-HT2A and 5-HT2C receptor inverse agonist with a hERG inhibitions, thus avoiding cardiovascular risks. 5-HT2A/5-HT2C inverse agonist 1 shows significant antipsychotic efficacy in the MK-801 (HY-15084B)-induced mouse model. 5-HT2A/5-HT2C inverse agonist 1 is promising for research of psychosis[1].
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5-HT2A/5-HT2C inverse agonist 1 | 5-HT2A/5-HT2C inverse agonist 1 is a potent and dual 5-HT2A and 5-HT2C receptor inverse agonist with a hERG inhibitions, thus avoiding cardiovascular risks. 5-HT2A/5-HT2C inverse agonist 1 shows significant antipsychotic efficacy in the MK-801 (HY-15084B)-induced mouse model. 5-HT2A/5-HT2C inverse agonist 1 is promising for research of psychosis. | |||||||||||||||||||||
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References
Keywords
