3011713-80-4
3011713-80-4
Chemical Structure
RSK-IN-2
- CAS No.: 3011713-80-4
- Formula:C25H30ClN7O3
- Molecular Weight:512.00
SMILES: CN1CCN(C2=CC(OC)=C(NC3=NC(NC4=CC=CC=C4C(NCCO)=O)=C(Cl)C=N3)C=C2)CC1
Biological Activity: RSK-IN-2 (Compound 3e) is a RSK inhibitor, with IC50 s of 37.89 nM (RSK2), 30.78 nM (RSK1), 20.51 nM (RSK3), 91.28 nM (RSK4). RSK-IN-2 inhibits tumor cell proliferation, induces apoptosis and causes cell cycle arrest in the G2/M phase[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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RSK-IN-2 | 99.32% | RSK-IN-2 (Compound 3e) is a RSK inhibitor, with IC50 s of 37.89 nM (RSK2), 30.78 nM (RSK1), 20.51 nM (RSK3), 91.28 nM (RSK4). RSK-IN-2 inhibits tumor cell proliferation, induces apoptosis and causes cell cycle arrest in the G2/M phase. | ||||||||||||||||||||
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References
Keywords
