3053862-47-5
3053862-47-5
Chemical Structure
FABP4-IN-3
- CAS No.: 3053862-47-5
- Formula:C20H16ClNO2
- Molecular Weight:337.80
InChIKey: RETKATZYCRROBY-UHFFFAOYSA-N
SMILES: O=C(C1=C(C)C=CC=C1NC2=C(C3=CC=CC=C3)C(Cl)=CC=C2)O
Biological Activity: FABP4-IN-3 (compound C3) is a highly selective FABP4 inhibitor (FABP4 Ki = 25 ± 3a nM, FABP3 Ki = 15.03 μM) which exhibits a 601-fold selectivity over FABP3. FABP4-IN-3 also shows metabolic stability and potent cellular anti-inflammatory activity, making it promising to get involved in the research of metabolic disease, cardiac dysfunction and inflammation-related disease[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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FABP4-IN-3 | 99.64% | FABP4-IN-3 (compound C3) is a highly selective FABP4 inhibitor (FABP4 Ki = 25 ± 3a nM, FABP3 Ki = 15.03 μM) which exhibits a 601-fold selectivity over FABP3. FABP4-IN-3 also shows metabolic stability and potent cellular anti-inflammatory activity, making it promising to get involved in the research of metabolic disease, cardiac dysfunction and inflammation-related disease. | ||||||||||||||||||||
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References
Keywords
