823817-56-7
823817-56-7
Chemical Structure
(Rac)-Sitagliptin
Synonym(s): (Rac)-MK-0431
- CAS No.: 823817-56-7
- Formula:C16H15F6N5O
- Molecular Weight:407.31
IUPAC Name: 3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)-4-(2,4,5-trifluorophenyl)butan-1-one
InChIKey: MFFMDFFZMYYVKS-UHFFFAOYSA-N
SMILES: O=C(N1CC2=NN=C(C(F)(F)F)N2CC1)CC(N)CC3=CC(F)=C(F)C=C3F
Biological Activity: (Rac)-Sitagliptin is an isoform of Sitagliptin (HY-13749), which is a potent and orally active inhibitor of DPP4 with an IC50 of 19 nM in Caco-2 cell extracts[1].
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(Rac)-Sitagliptin | (Rac)-Sitagliptin is an isoform of Sitagliptin (HY-13749), which is a potent and orally active inhibitor of DPP4 with an IC50 of 19 nM in Caco-2 cell extracts. | |||||||||||||||||||||
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References
Keywords
