2. Metabolic Enzyme/Protease
  3. Endogenous Metabolite
  4. MRS2802

MRS2802 is a P2Y14 receptor agonist with an EC50 value of 63 nM. MRS2802 can effectively activate the P2Y14 receptor and may play a role in regulating platelet function. The selectivity and activity of MRS2802 are conducive to in-depth research on the biological functions and pharmacological properties of P2Y receptors. The development of MRS2802 provides a potential inhibitory strategy for the search for new antiplatelet compounds.

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MRS2802

MRS2802 화학구조

CAS No. : 1047980-53-9

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MRS2802 Related Antibodies

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제품 설명

MRS2802 is a P2Y14 receptor agonist with an EC50 value of 63 nM. MRS2802 can effectively activate the P2Y14 receptor and may play a role in regulating platelet function. The selectivity and activity of MRS2802 are conducive to in-depth research on the biological functions and pharmacological properties of P2Y receptors. The development of MRS2802 provides a potential inhibitory strategy for the search for new antiplatelet compounds[1].

Cellular Effect
Cell Line Type Value Description References
HEK293 EC50
63 nM
Compound: 12
Agonist activity at human P2Y14 receptor expressed in HEK293 cells coexpressing phospholipase C-activating Gi protein cells assessed as inhibition of forskolin induced [3H]cAMP production
Agonist activity at human P2Y14 receptor expressed in HEK293 cells coexpressing phospholipase C-activating Gi protein cells assessed as inhibition of forskolin induced [3H]cAMP production
[PMID: 19902968]
분자량

438.17

화학식

C10H14F2N2O11P2
CAS No.
SMILES

O=C(C=CN1[C@@H]2O[C@H](COP(O)(C(P(O)(O)=O)(F)F)=O)[C@@H](O)[C@H]2O)NC1=O
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
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MRS2802 Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

MRS28021047980-53-9MRS 2802MRS-2802Endogenous MetaboliteInhibitorinhibitorinhibit

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상품명:
MRS2802
Cat. No.:
HY-122211
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