Opioid receptor agonist 1
Opioid receptor agonist 1 (Compound 2638-28) is the orally active agonist for opioid receptor that exhibits good affinity to MOR, DOR and KOR with Ki of 5, 24 and 212 nM, respectively. Opioid receptor agonist 1 exhibits analgesic activity in mouse warm water tail flick models and acetic acid writhing models.
For research use only. We do not sell to patients.
- Formula: C32H45N5O
- Molecular Weight:515.73
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Opioid Receptor Isoforms
More
Biological Activity
|
μ Opioid Receptor/MOR 5 nM (Ki) |
δ Opioid Receptor/DOR 24 nM (Ki) |
κ Opioid Receptor/KOR 212 nM (Ki) |
Chemical Information
-
Molecular Weight 515.73
-
Formula C32H45N5O
-
SMILES
CC(C)C[C@H]1CN2[C@@H](CC3=CC=C(O)C=C3)CN4[C@@H](CCN(C)C)CN=C4C=C2N1CCC5=CC=CC=C5
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)