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Pitavastatin-d4 hemicalcium

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "Pitavastatin-d4 hemicalcium" in MCE Product Catalog:

Cat. No.: HY-B0144S
Synonyms: NK-104-d4 hemicalcium; Pitavastatin-d4 hemicalcium
Pitavastatin-d4 (hemicalcium) is deuterium labeled Pitavastatin (Calcium). Pitavastatin Calcium (NK-104 hemicalcium) is a potent hydroxymethylglutaryl-CoA (HMG-CoA) reductase inhibitor. Pitavastatin Calcium (NK-104 hemicalcium) inhibits cholesterol synthesis from acetic acid with an IC50 of 5.8 nM in HepG2 cells. Pitavastatin Calcium is an efficient hepatocyte low-density lipoprotein-cholesterol (LDL-C) receptor inducer. Anti-cancer activity[1][2][3].
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