3 Results for "

Androgen receptor-IN-7

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "Androgen receptor-IN-7" in MCE Product Catalog:

Cat. No.: HY-179050
CAS No.: 401580-43-6
Research Areas:  

Cancer

Androgen receptor-IN-7 is a potent androgen receptor (AR) inhibitor. Androgen receptor-IN-7 exhibits potent anticancer activity against PC-3 cells (IC50 =370.37 nM) and LNCaP cells via both AR-dependent and AR-independent pathways. Androgen receptor-IN-7 induces ROS production in PC-3 cells. Androgen receptor-IN-7 can be used for prostate cancer research .
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Cat. No.: HY-110028
CAS No.: 16496-99-4
Purity:  99.06%
Leelamine hydrochloride is an orally active weakly basic amine that inhibits NPC1 and the androgen receptor AR-V7, and acts as a cannabinoid receptor agonist. Leelamine hydrochloride also functions as a lysosome affinity agent that blocks endocytosis, disrupts autophagic flux and cholesterol transport, thereby altering the RTK-AKT/STAT/MAPK signaling cascade. Leelamine hydrochloride induces cancer cell death and autophagosome accumulation, and can be used in research related to melanoma, castration-resistant prostate cancer and breast cancer .
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Cat. No.: HY-152524
CAS No.: 2409791-89-3
Target:  

Androgen Receptor

Research Areas:  

Cancer

Androgen receptor antagonist 7 is an effective androgen receptor (AR) antagonist with an IC50 value of 1.18 µM. Androgen receptor antagonist 7 has biological activity in vitro and inhibits the expression of AR target in a time and dose dependent manner with an GI50 value of 7.9 µM .
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