16 Results for "

Fesoterodine fumarate

" in MedChemExpress (MCE) Product Catalog:
Products (16)

16 Results for "Fesoterodine fumarate" in MCE Product Catalog:

Cat. No.: HY-A0030
CAS No.: 286930-03-8
Target:  

mAChR

Fesoterodine Fumarate is an orally active, nonsubtype selective, competitive muscarinic receptor (mAChR) antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. Fesoterodine Fumarate is used for the overactive bladder (OAB) .
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1 Cited Publications
Cat. No.: HY-76569
CAS No.: 207679-81-0
Synonyms: PNU-200577; 5-Hydroxymethyl Tolterodine
Target:  

mAChR

Research Areas:  

Neurological Disease Cancer

Desfesoterodine (PNU-200577) is a potent and selective muscarinic receptor (mAChR) antagonist with a KB and a pA2 of 0.84 nM and 9.14, respectively . Desfesoterodine is a major pharmacologically active metabolite of Tolterodine (PNU-200583; HY-A0024) and Fesoterodine (HY-70053) . Desfesoterodine improves cerebral infarction induced detrusor overactivity in rats .
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Cat. No.: HY-70053
CAS No.: 286930-02-7
Target:  

mAChR

Fesoterodine is an orally active, nonsubtype selective, competitive muscarinic receptor (mAChR) antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. Fesoterodine is used for the overactive bladder (OAB) .
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Cat. No.: HY-70053A
CAS No.: 1206695-46-6
Target:  

mAChR

Fesoterodine L-mandelate is an orally active, nonsubtype selective, competitive muscarinic receptor (mAChR) antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. Fesoterodine L-mandelate is used for the overactive bladder (OAB) .
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Cat. No.: HY-A0030S
CAS No.: 2747918-94-9
Fesoterodine-d7 (fumarate) is the deuterium labeled Fesoterodine fumarate . Fesoterodine Fumarate is an orally active, nonsubtype selective, competitive muscarinic receptor (mAChR) antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. Fesoterodine Fumarate is used for the overactive bladder (OAB) .
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Cat. No.: HY-W720879
CAS No.: 1126611-84-4
Fesoterodine-d3 is the deuterium labeled Fesoterodine (HY-70053). Fesoterodine is an orally active, nonsubtype selective, competitive muscarinic receptor (mAChR) antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. Fesoterodine is used for the overactive bladder (OAB) .
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Cat. No.: HY-A0030R
CAS No.: 286930-03-8
Fesoterodine (fumarate) (Standard) is the analytical standard of Fesoterodine (fumarate). This product is intended for research and analytical applications. Fesoterodine Fumarate is an orally active, nonsubtype selective, competitive muscarinic receptor (mAChR) antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. Fesoterodine Fumarate is used for the overactive bladder (OAB) .
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Cat. No.: HY-43452S
CAS No.: 2747918-96-1
Fesoterodine-d7 (hydrochloride) is deuterium labeled 2-(3-(Diisopropylamino)-1-phenylpropyl)-4-(hydroxymethyl)phenyl isobutyrate.
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Cat. No.: HY-70053S
CAS No.: 1185237-08-4
(Rac)-Fesoterodine-d14 fumarate is a labelled racemic Fesoterodine. Fesoterodine is an orally active, nonsubtype selective, competitive muscarinic receptor (mAChR) antagonist with pKivalues of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. Fesoterodine is used for the overactive bladder (OAB) .
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Cat. No.: HY-76569R
CAS No.: 207679-81-0
Synonyms: PNU-200577 (Standard); 5-Hydroxymethyl Tolterodine (Standard)
Research Areas:  

Neurological Disease

Desfesoterodine (Standard) is the analytical standard of Desfesoterodine. This product is intended for research and analytical applications. Desfesoterodine (PNU-200577) is a potent and selective muscarinic receptor (mAChR) antagonist with a KB and a pA2 of 0.84 nM and 9.14, respectively . Desfesoterodine is a major pharmacologically active metabolite of Tolterodine (PNU-200583; HY-A0024) and Fesoterodine (HY-70053) . Desfesoterodine improves cerebral infarction induced detrusor overactivity in rats .
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Cat. No.: HY-76569B
CAS No.: 380636-49-7
Synonyms: PNU-200577 formic
Target:  

mAChR

Research Areas:  

Neurological Disease

5-Hydroxymethyl tolterodine (formate) (PNU-200577 (formic)) is an active metabolite of the muscarinic acetylcholine receptor antagonists Tolterodine (HY-A0024) and Fesoterodine (HY-70053). 5-Hydroxymethyl tolterodine (formate) is formed from tolterodine by the cytochrome P450 (CYP) isoform CYP2D6 and from fesoterodine by plasma esterases.
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Cat. No.: HY-180471
CAS No.: 1361197-33-2
Target:  

Drug Metabolite

Research Areas:  

Others

Desisopropyl-fesoterodine (compound 1), an oxidative Ndealkylation of the tertiary amine function of Fesoterodine (HY-70053), is a degradation product (compound PP-6) of Fesoterodine .
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Cat. No.: HY-I0104
CAS No.: 250214-69-8
Target:  

Drug Intermediate

Research Areas:  

Others

Fesoterodine impurity 1 is an impurity of Fesoterodine (HY-70053).
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Cat. No.: HY-76569S1
CAS No.: 1191280-58-6
Synonyms: PNU-200577-d14; 5-Hydroxymethyl Tolterodine-d14
(R)-Hydroxytolterodine-d14 is deuterated labeled Desfesoterodine (HY-76569). Desfesoterodine (PNU-200577) is a potent and selective muscarinic receptor (mAChR) antagonist with a KB and a pA2 of 0.84 nM and 9.14, respectively . Desfesoterodine is a major pharmacologically active metabolite of Tolterodine (PNU-200583; HY-A0024) and Fesoterodine (HY-70053) . Desfesoterodine improves cerebral infarction induced detrusor overactivity in rats .
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Cat. No.: HY-I0104R
CAS No.: 250214-69-8
Target:  

Reference Standards

2-[3-[Bis(1-methylethyl)amino]-1-phenylpropyl]-4-(methoxymethyl)phenol (Standard) is the analytical standard of 2-[3-[Bis(1-methylethyl)amino]-1-phenylpropyl]-4-(methoxymethyl)phenol. This product is intended for research and analytical applications.
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Cat. No.: HY-76569S
Synonyms: PNU-200577-d5; 5-Hydroxymethyl Tolterodine-d5
Desfesoterodine-d5 (PNU-200577-d5) is the deuterium labeled Desfesoterodine (HY-76569). Desfesoterodine (PNU-200577) is a potent and selective muscarinic receptor (mAChR) antagonist with a KB and a pA2 of 0.84 nM and 9.14, respectively . Desfesoterodine is a major pharmacologically active metabolite of Tolterodine (PNU-200583; HY-A0024) and Fesoterodine (HY-70053) . Desfesoterodine improves cerebral infarction induced detrusor overactivity in rats .
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