country

Change Language

EN - English
FR - Français
DE - Deutsch
ES - Español
JA - 日本語
KO - 한국어

Country or Region:

United States

Product Name	Size / Unit Price	Qty

Total: USD 0.00 Checkout

Cat. No.: HY-76569B

Copy Link Print Information

5-Hydroxymethyl tolterodine formate

Name: 5-Hydroxymethyl tolterodine formate
Brand: MedChemExpress
SKU: HY-76569B
Availability: PreOrder

(Synonyms: PNU-200577 formic)

1 Cited Publications

Customer Review

Based on 1 publication(s) in Google Scholar

5-Hydroxymethyl tolterodine (formate) (PNU-200577 (formic)) is an active metabolite of the muscarinic acetylcholine receptor antagonists Tolterodine (HY-A0024) and Fesoterodine (HY-70053). 5-Hydroxymethyl tolterodine (formate) is formed from tolterodine by the cytochrome P450 (CYP) isoform CYP2D6 and from fesoterodine by plasma esterases.

For research use only. We do not sell to patients.

CAS No.: 380636-49-7
Formula: C₂₃H₃₃NO₄
Molecular Weight:387.51

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (268 KB)

5-Hydroxymethyl tolterodine formate Chemical Structure

CAS No.: 380636-49-7

Size

Price

Stock

Quantity

Amount: USD 0.00

* Please select Quantity before adding items.

Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

All mAChR Isoforms :

Chemical Information

CAS No. 380636-49-7
Molecular Weight 387.51
Formula C₂₃H₃₃NO₄
SMILES

OC1=C(C=C(CO)C=C1)[C@@H](C2=CC=CC=C2)CCN(C(C)C)C(C)C.OC=O
Synonyms

PNU-200577 formic
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Publications (1)

All

Sort by:

Journal Impact Factor

Sci Rep

Tolterodine is a novel candidate for assessing CYP3A4 activity through metabolic volatiles to predict drug responses. [Abstract]

2025 Jan 20;15(1):2462. PMID: 39828876

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (268 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. L Nilvebrant, et al. Antimuscarinic potency and bladder selectivity of PNU-200577, a major metabolite of tolterodine. Pharmacol Toxicol. 1997 Oct;81(4):169-72. [Content Brief]

Calculators

Molarity Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Dilution Calculator

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

Keywords

5-Hydroxymethyl tolterodine formate

1 Cited Publications

100 mg Get Quote

Subscribe to the

MedChemExpress

Newsletter

MOQ

Minimum order quantity

100 mg

Get Quote In-stock

Other size

Get Quote

Amount: USD 0.00

Biological Activity
- Description
Chemical Information
Publications (1)
Purity & Documentation
References

Product Name:
Cat. No.:
Quantity:
MCE Japan Authorized Agent:

Product Name:
CAS No.:
Species:
Purity:
Quantity:

5-Hydroxymethyl tolterodine formate

FB23

5-Hydroxyomeprazole

Pantoprazole sulfide

Lansoprazole sulfone

2'-C-Methylguanosine

2-(1-Piperazinyl)pyrimidine

Lansoprazole sulfone (Standard)

2-(1-Piperazinyl)pyrimidine (Standard)

5-Hydroxyomeprazole (Standard)

Pantoprazole sulfone

10-Hydroxywarfarin

3-Hydroxyquinine

Publications Citing Use of MedChemExpress (MCE) 5-Hydroxymethyl tolterodine formate

All mAChR Isoforms

Biological Activity

Chemical Information

Publications (1)

Purity & Documentation

References

Calculators

Help & FAQs

Bioz

5-Hydroxymethyl tolterodine formate

FB23

5-Hydroxyomeprazole

Pantoprazole sulfide

Lansoprazole sulfone

2'-C-Methylguanosine

2-(1-Piperazinyl)pyrimidine

Lansoprazole sulfone (Standard)

2-(1-Piperazinyl)pyrimidine (Standard)

5-Hydroxyomeprazole (Standard)

Pantoprazole sulfone

10-Hydroxywarfarin

3-Hydroxyquinine

Publications Citing Use of MedChemExpress (MCE) 5-Hydroxymethyl tolterodine formate

All mAChR Isoforms

Biological Activity

Chemical Information

Publications (1)

Purity & Documentation

References

Calculators

Help & FAQs

5-Hydroxymethyl tolterodine formate Related Classifications

HY-76569B Related Classifications

Bioz