1 Result for "

I-BET282E

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "I-BET282E" in MCE Product Catalog:

Cat. No.: HY-19760B
CAS No.: 2885162-99-0
Research Areas:  

Inflammation/Immunology

I-BET282E is a pan-inhibitor of all eight BET bromodomains, and selectivity over other representative bromodomain-containing proteins. I-BET282E shows pIC50s ranging 6.4-7.7 for BRD2 (BD1/BD2), BRD2 (BD1/BD), BRD3 (BD1/BD), and BRD4 (BD1/BD) .
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