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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
13 Results for "
Leu-enkephalin
" in MedChemExpress (MCE) Product Catalog:
Products (13)
13 Results for "Leu-enkephalin" in MCE Product Catalog:
2
2 Cited Publications
Cat. No.: HY-P0288
CAS No.: 58822-25-6
Synonyms: Leu-enkephalin; Leucine enkephalin; Leucyl-enkephalin
Target:
Cat. No.: HY-P1170
CAS No.: 2703746-32-9
Synonyms: Ac-L-Tyr-Gly-Gly-L-Phe-D-Leu-COOH
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Cat. No.: HY-W009602
CAS No.: 3918-87-4
Synonyms: Phe-ala
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Cat. No.: HY-P0098
CAS No.: 64963-01-5
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Cat. No.: HY-P1470
CAS No.: 60117-24-0
Synonyms: Leu-enkephalin amide
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BMS-986187 is an δ-opioid receptor-selective positive allosteric modulator (PAM) with an EC50 of 0.03 μM and a pKB of 6.02 (～1 μM). BMS-986187 has no observable PAM activity at the μ-receptor (EC50=3 μM) .
Cat. No.: HY-P3513
CAS No.: 77739-21-0
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Cat. No.: HY-115500
CAS No.: 1206514-50-2
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PL265 is an orally active dual enkephalinase inhibitor. PL265 is a prodrug of PL254, which can simultaneously and efficiently inhibit neutral endopeptidase (Neprilysin) and Aminopeptidase N. PL265 can effectively protect and significantly increase the local concentration of enkephalins (such as Met-Enkephalin and Leu-Enkephalin) released by cells at the pain or inflammation sites, thereby activating μ and δ opioid receptors to produce a potent analgesic effect. PL254 can also inhibit leukotriene A4 hydrolase (LTA4H), which may contribute to its additional anti-inflammatory effect by reducing the production of pro-inflammatory mediator leukotriene B4 (LTB4). PL265 can be used in non-addictive chronic pain research .
Cat. No.: HY-106975
CAS No.: 144505-58-8
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SCH-42354 is a potent, orally active neutral endopeptidase (NEP) inhibitor, is the pharmacologically active form of the proagent SCH-42495. SCH-42354 inhibits the hydrolysis of NEP to enhance the activity of atrial natriuretic peptide (ANP). SCH-42354 inhibits hydrolysis of leu-enkephalin and ANF with IC50 values of 8.3 nM and 10.0 nM, respectively. SCH-42354 has antihypertensive activity .
Cat. No.: HY-W009602R
CAS No.: 3918-87-4
Synonyms: Phe-ala (Standard)
Cat. No.: HY-P3513A
CAS No.: 78658-39-6
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β-Neo-Endorphin acetate is an endogenous opioid peptide. β-Neo-Endorphin acetate is a hypothalamic "big" Leu-enkephalin of porcine origin. β-Neo-Endorphin acetate shows activation of the Erk1/2, MMP-2 and MMP-9 .
Cat. No.: HY-P71058
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: PDYN; Neoendorphin-Dynorphin-enkephalin Prepropeptide; Prev. SCA23; Leu-enkephalin; Beta-Neoendorphin-Dynorphin; Leumorphin; Proenkephalin-B; Rimorphin; Preprodynorphin; Spinocerebellar Ataxia 23; PENKB; Beta-Neoendorphin; ADCA; Dynorphin; Prodynorphin; P
Species:
Human
Source:
HEK293
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
