1 Result for "

Leucettinib 92

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "Leucettinib 92" in MCE Product Catalog:

Cat. No.: HY-155723
CAS No.: 2732859-57-1
Purity:  98.54%
Target:  

CDK DYRK

Research Areas:  

Others

Leucettinib-92 (compound 92) is an inhibitor of DYRK/CLK kinase, The IC50s are 147 nM (CLK1), 39 nM (CLK2), 5.2 nM (CLK4), 0.8 μM (CLK3), 124 nM (DYRK1A), 204 nM (DYRK1B), 0.16 μM (DYRK2), respectively. 1.0 μM (DYRK3), 0.52 μM (DYRK4), 2.78 μM (GSK3) .
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