2 Results for "

Naltrindole hydrochloride

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Naltrindole hydrochloride" in MCE Product Catalog:

Cat. No.: HY-136208
CAS No.: 892039-23-5
Purity:  99.44%
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

TAN-452 is an orally active, selective peripherally acting δ-opioid receptor (DOR) antagonist with a Ki of 0.47 nM and a Kb of 0.21 nM. TAN-452 is an antagonist for μ-opioid receptor (MOR; Ki=36.56 nM and Kb=9.43 nM) and κ-opioid receptor (KOR; Ki=5.31 nM and Kb=7.18 nM). TAN-452, a derivative of Naltrindole, demonstrates low brain penetrability and attenuates morphine-induced side effects without affecting pain control .
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Cat. No.: HY-172149
CAS No.: 126876-64-0
Synonyms: 5'-NTII
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Naltrindole 5′-isothiocyanate (5'-NTII) is a non-selective delta opioid receptor antagonist that can antagonize the analgesic effects induced by DSLET (HY-P1332) without affecting the analgesic effects induced by DPDPE (HY-P1334) .
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