1 Result for "

PROTAC ITK degrader 1

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "PROTAC ITK degrader 1" in MCE Product Catalog:

Cat. No.: HY-149917
Target:  

PROTACs Itk

Research Areas:  

Cancer

PROTAC ITK degrader 1 is a highly selective degrader of interleukin-2-inducible T-cell kinase (ITK; DC50=3.6 nM in vivo in mice), with good plasma exposure levels. PROTAC ITK degrader 1 induces rapid, and prolonged ITK degradation and suppresses IL-2 secretion (EC50=35.2 nM, Jurkat cells) stimulated by anti-CD3 antibodyin vivo .
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