1 Result for "

RVD-Hpα TFA

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "RVD-Hpα TFA" in MCE Product Catalog:

Art. -Nr.: HY-P1397A
CAS. Nr.: 1431329-51-9
Target:  

Cannabinoid Receptor

Forschungsgebiete:  

Cardiovascular Disease

RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca 2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM).
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