1 Result for "

Umbralisib sulfate

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "Umbralisib sulfate" in MCE Product Catalog:

Cat. No.: HY-12279B
CAS No.: 1532533-75-7
Synonyms: TGR-1202 sulfate; RP-5264 sulfate
Target:  

PI3K Casein Kinase

Research Areas:  

Cancer

Umbralisib (TGR-1202) sulfate is an orally active, potent and selective dual PI3Kδ and casein kinase-1-ε (CK1ε) inhibitor, with EC50 of 22.2 nM and 6.0 μM, respectively. Umbralisib sulfate exhibits unique immunomodulatory effects on chronic lymphocytic leukemia (CLL) T cells. Umbralisib sulfate can be used for haematological malignancies reseach .
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