3 Results for "

direct PDK1 inhibitor

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "direct PDK1 inhibitor" in MCE Product Catalog:

7
7 Cited Publications
Cat. No.: HY-11005
CAS No.: 702674-56-4
Purity:  99.13%
Target:  

PDK-1 Apoptosis

Research Areas:  

Cancer

BX-912 is a direct, selective, and ATP-competitive PDK1 inhibitor (IC50=26 nM). BX-912 blocks PDK1/Akt signaling in tumor cells and inhibits the anchorage-dependent growth of a variety of tumor cell lines in culture or induces apoptosis .
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Cat. No.: HY-10515
CAS No.: 702676-93-5
Purity:  99.4%
Target:  

PDK-1

Research Areas:  

Cancer

BX-320 is a selective, ATP-competitive, orally acitive, and direct PDK1 inhibitor with an IC50 of 30 nM in a direct kinase assay format. BX-320 also induces apoptosis. Anticancer effect .
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Cat. No.: HY-11005R
CAS No.: 702674-56-4
Research Areas:  

Cancer

BX-912 (Standard) is the analytical standard of BX-912 (HY-11005). This product is intended for research and analytical applications. BX-912 is a direct, selective, and ATP-competitive PDK1 inhibitor (IC50=26 nM). BX-912 blocks PDK1/Akt signaling in tumor cells and inhibits the anchorage-dependent growth of a variety of tumor cell lines in culture or induces apoptosis .
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