1609522-33-9
1609522-33-9
Chemical Structure
SEL120-34A
- CAS No.: 1609522-33-9
- Formula:C15H18Br2N4
- Molecular Weight:414.14
IUPAC Name: 7,8-dibromo-9-methyl-2-(piperazin-1-yl)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinoline
InChIKey: FSBMCTDYWXIBLM-UHFFFAOYSA-N
SMILES: CC1=C2C3=C(C(Br)=C1Br)CCCN3C(N4CCNCC4)=N2
Biological Activity: SEL120-34A is a potent, selective, orally available, ATP-competitive CDK8 inhibitor, with IC50s of 4.4 nM and 10.4 nM for CDK8/CycC and CDK19/CycC, respectively, with antitumor activity.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
SEL120-34A | 99.49% | SEL120-34A is a potent, selective, orally available, ATP-competitive CDK8 inhibitor, with IC50s of 4.4 nM and 10.4 nM for CDK8/CycC and CDK19/CycC, respectively, with antitumor activity. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
