2468783-22-2
2468783-22-2
Chemical Structure
BJP-07-017-3
- CAS No.: 2468783-22-2
- Formula:C35H45ClN8O6
- Molecular Weight:709.23
InChIKey: CGODJOIFYRVRID-DZUOILHNSA-N
SMILES: CN(C(CCl)=O)[C@H](C(N1CCCC[C@H]1C(N[C@H](C(N[C@@H](CCCNC(N)=O)C(N)=O)=O)CC2=CNC3=C2C=CC=C3)=O)=O)CC4=CC=CC=C4
Biological Activity: BJP-07-017-3 is the inhibitor for proline cis trans isomerase (Pin1) with an IC50 of 9 nM. BJP-07-017-3 forms covalent bond with Cys113 of Pin1, induces conformational changes in Pin1, reduces its stability, and leads to a proteasome-dependently degradation[1].
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BJP-07-017-3 | BJP-07-017-3 is the inhibitor for proline cis trans isomerase (Pin1) with an IC50 of 9 nM. BJP-07-017-3 forms covalent bond with Cys113 of Pin1, induces conformational changes in Pin1, reduces its stability, and leads to a proteasome-dependently degradation. | |||||||||||||||||||||
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