CDK2/9-IN-1
CDK2/9-IN-1 (compound 20a) is an orally active dual inhibitor of CDK2 and CDK9 with IC50 values are 0.004 μM and 0.009 μM respectively. CDK2/9-IN-1 induces apoptosis by regulating G2/M cell cycle arrest. CDK2/9-IN-1 has antitumor activity.
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- CAS No.: 2222285-23-4
- Formule: C14H14N6O2S2
- Masse moléculaire:362.43
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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CDK2 0.004 μM (IC50) |
CDK9 0.009 μM (IC50) |
Chemical Information
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CAS No. 2222285-23-4
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Masse moléculaire 362.43
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Formule C14H14N6O2S2
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SMILES
O=S(C1=CC=C(NC2=NC(NC3=NC=CS3)=C(C=N2)C)C=C1)(N)=O
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)