2222285-23-4
2222285-23-4
Chemical Structure
CDK2/9-IN-1
- CAS No.: 2222285-23-4
- Formula:C14H14N6O2S2
- Molecular Weight:362.43
SMILES: O=S(C1=CC=C(NC2=NC(NC3=NC=CS3)=C(C=N2)C)C=C1)(N)=O
Biological Activity: CDK2/9-IN-1 (compound 20a) is an orally active dual inhibitor of CDK2 and CDK9 with IC50 values are 0.004 μM and 0.009 μM respectively. CDK2/9-IN-1 induces apoptosis by regulating G2/M cell cycle arrest. CDK2/9-IN-1 has antitumor activity[1].
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CDK2/9-IN-1 | CDK2/9-IN-1 (compound 20a) is an orally active dual inhibitor of CDK2 and CDK9 with IC50 values are 0.004 μM and 0.009 μM respectively. CDK2/9-IN-1 induces apoptosis by regulating G2/M cell cycle arrest. CDK2/9-IN-1 has antitumor activity. | |||||||||||||||||||||
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References
Keywords
