111205-55-1
Chemical Structure
CGS 20625
- CAS No.: 111205-55-1
- Formula:C18H19N3O2
- Molecular Weight:309.36
IUPAC Name: 2-(4-methoxyphenyl)-5,6,7,8,9,10-hexahydrocyclohepta[b]pyrazolo[3,4-d]pyridin-3(2H)-one
InChIKey: XRUUVUYJUULCBQ-UHFFFAOYSA-N
SMILES: O=C1C2=CNC(CCCCC3)=C3C2=NN1C4=CC=C(OC)C=C4
Biological Activity: CGS 20625 is a potent, selective and orally active partial agonist for the central benzodiazepine receptor. CGS 20625 inhibits [3H]-flunitrazepam binding to central benzodiazepine receptors with an IC50 of 1.3 nM. CGS 20625 enhances GABA in Xenopus laevis oocytes . CGS 20625 can be used for the research of pentylenetetrazol-induced seizures and anxiety[1][2].
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CGS 20625 | 99.80% | CGS 20625 is a potent, selective and orally active partial agonist for the central benzodiazepine receptor. CGS 20625 inhibits [3H]-flunitrazepam binding to central benzodiazepine receptors with an IC50 of 1.3 nM. CGS 20625 enhances GABA in Xenopus laevis oocytes . CGS 20625 can be used for the research of pentylenetetrazol-induced seizures and anxiety. | ||||||||||||||||||||
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Keywords
