1197824-15-9
1197824-15-9
Chemical Structure
EN4
- CAS No.: 1197824-15-9
- Formula:C25H24N2O4
- Molecular Weight:416.47
IUPAC Name: 4-(acrylamidomethyl)-N-(2-(4-ethoxyphenoxy)phenyl)benzamide
InChIKey: DKOWGKKELPCHEG-UHFFFAOYSA-N
SMILES: O=C(NC1=CC=CC=C1OC2=CC=C(OCC)C=C2)C3=CC=C(CNC(C=C)=O)C=C3
Biological Activity: EN4 is a covalent ligand that targets cysteine 171 (C171) of MYC. EN4 is selective for c-MYC over N-MYC and L-MYC. EN4 inhibits MYC transcriptional activity, downregulates MYC targets, and impairs tumorigenesis[1].
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EN4 | 96.29% | EN4 is a covalent ligand that targets cysteine 171 (C171) of MYC. EN4 is selective for c-MYC over N-MYC and L-MYC. EN4 inhibits MYC transcriptional activity, downregulates MYC targets, and impairs tumorigenesis. | ||||||||||||||||||||
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