1232221-74-7
Chemical Structure
APY0201
- CAS No.: 1232221-74-7
- Formula:C23H23N7O
- Molecular Weight:413.48
IUPAC Name: (E)-4-(5-(2-(3-methylbenzylidene)hydrazinyl)-2-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl)morpholine
InChIKey: RFZQYGBLRIKROZ-PCLIKHOPSA-N
SMILES: CC1=CC(/C=N/NC2=NC3=CC(C4=CC=NC=C4)=NN3C(N5CCOCC5)=C2)=CC=C1
Biological Activity: APY0201 is a potent PIKfyve inhibitor, which inhibits the conversion of PtdIns3P to PtdIns(3,5)P2 in the presence of in the presence of [33P]ATP with an IC50 of 5.2 nM. APY0201 also inhibits IL-12/IL-23 production.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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APY0201 | 99.42% | APY0201 is a potent PIKfyve inhibitor, which inhibits the conversion of PtdIns3P to PtdIns(3,5)P2 in the presence of in the presence of [33P]ATP with an IC50 of 5.2 nM. APY0201 also inhibits IL-12/IL-23 production. | ||||||||||||||||||||
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Keywords