1332708-14-1
Chemical Structure
PF-4840154
- CAS No.: 1332708-14-1
- Formula:C26H38N6O2
- Molecular Weight:466.62
IUPAC Name: N-benzyl-4-(isobutylamino)-2-(4-((tetrahydro-2H-pyran-3-yl)methyl)piperazin-1-yl)pyrimidine-5-carboxamide
InChIKey: PPANZCQXFYBGHN-UHFFFAOYSA-N
SMILES: O=C(C1=CN=C(N2CCN(CC3COCCC3)CC2)N=C1NCC(C)C)NCC4=CC=CC=C4
Biological Activity: PF-4840154 is a potent, selective agonist of the rat and human TrpA1 channel with EC50s of 97 and 23 nM, respectively. PF-4840154 elicits TrpA1-mediated nocifensive behaviour in mouse[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PF-4840154 | 98.15% | PF-4840154 is a potent, selective agonist of the rat and human TrpA1 channel with EC50s of 97 and 23 nM, respectively. PF-4840154 elicits TrpA1-mediated nocifensive behaviour in mouse. | ||||||||||||||||||||
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Keywords