148440-81-7
148440-81-7
Chemical Structure
Thioperamide maleate
Synonym(s): MR-12842 maleate
- CAS No.: 148440-81-7
- Formula:C15H24N4S.xC4H4O4
- Molecular Weight:N/A
SMILES: S=C(N1CCC(C2=CN=CN2)CC1)NC3CCCCC3.O=C(O)/C=C\C(O)=O.[x]
Biological Activity: Thioperamide maleate (MR-12842 maleate) is a potent, orally available, brain penetrant and selective H3 receptor antagonist with a Ki of 4.3 nM for inhibition of [3H]histamine release. Thioperamide maleate inhibits [3H]histamine synthesis with a Ki of 31 nM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Thioperamide maleate | 98.26% | Thioperamide maleate (MR-12842 maleate) is a potent, orally available, brain penetrant and selective H3 receptor antagonist with a Ki of 4.3 nM for inhibition of [3H]histamine release. Thioperamide maleate inhibits [3H]histamine synthesis with a Ki of 31 nM. | ||||||||||||||||||||
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References
Keywords
