151272-90-1
151272-90-1
Chemical Structure
CP-135807
- CAS No.: 151272-90-1
- Formula:C19H21N5O2
- Molecular Weight:351.40
IUPAC Name: (R)-3-((1-methylpyrrolidin-2-yl)methyl)-N-(3-nitropyridin-2-yl)-1H-indol-5-amine
InChIKey: YPFIYPNOWVPAPR-OAHLLOKOSA-N
SMILES: O=[N+](C1=CC=CN=C1NC2=CC3=C(NC=C3C[C@@H]4N(C)CCC4)C=C2)[O-]
Biological Activity: CP-135807 is an orally active and selective 5-HT1D agonist (IC50=3.1 nM), bovine). CP-135807 mediates central psychoactivity and can be used in antidepressant research[1][2].
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CP-135807 | CP-135807 is an orally active and selective 5-HT1D agonist (IC50=3.1 nM), bovine). CP-135807 mediates central psychoactivity and can be used in antidepressant research. | |||||||||||||||||||||
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References
- [1]. Mansbach RS, et al. CP-135,807, a selective 5-HT1D agonist: effects in drug discrimination and punishment procedures in the pigeon. Psychopharmacology (Berl). 1996 Dec;128(3):313-9. [Content Brief]
- [2]. Macor J E, et al. Use of 2, 5-Dimethylpyrrole as an Amino-Protecting Group in an Efficient Synthesis of 5-Amino-3-[(N-methyl-pyrrolidin-2 (R)-yl) methyl] indole[J]. The Journal of Organic Chemistry, 1994, 59(24): 7496-7498.
