1612158-07-2
1612158-07-2
Chemical Structure
DS43260857
- CAS No.: 1612158-07-2
- Formula:C19H16F3N3O3S
- Molecular Weight:423.41
InChIKey: IEMVZIXARQGLOW-UHFFFAOYSA-N
SMILES: CC1=CN(C2=CC(C(F)(F)F)=CN=C2)C3=C1C=C(C(NS(C4CC4)(=O)=O)=O)C=C3
Biological Activity: DS43260857 is a potentNaV1.7inhibitor, which has a high inhibitory effect on both human and mouse NaV1.7. The IC50 values of DS43260857 for hNaV1.1, hNaV1.5, hNaV1.7, mNaV1.7 are 6.6, 14, 0.015 and 0.061 μM, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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DS43260857 | 98.71% | DS43260857 is a potentNaV1.7inhibitor, which has a high inhibitory effect on both human and mouse NaV1.7. The IC50 values of DS43260857 for hNaV1.1, hNaV1.5, hNaV1.7, mNaV1.7 are 6.6, 14, 0.015 and 0.061 μM, respectively. | ||||||||||||||||||||
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References
Keywords
