1693758-51-8
1693758-51-8
Chemical Structure
Eganelisib
Synonym(s): IPI-549
- CAS No.: 1693758-51-8
- Formula:C30H24N8O2
- Molecular Weight:528.56
IUPAC Name: (S)-2-amino-N-(1-(8-((1-methyl-1H-pyrazol-4-yl)ethynyl)-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl)ethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
InChIKey: XUMALORDVCFWKV-IBGZPJMESA-N
SMILES: O=C(C1=C2N=CC=CN2N=C1N)N[C@H](C3=CC4=C(C(N3C5=CC=CC=C5)=O)C(C#CC6=CN(C)N=C6)=CC=C4)C
Biological Activity: Eganelisib (IPI549) is a potent and selective PI3Kγ inhibitor with an IC50 of 16 nM. Eganelisib shows >100-fold selectivity over other lipid and protein kinases[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Eganelisib | 99.68% | Eganelisib (IPI549) is a potent and selective PI3Kγ inhibitor with an IC50 of 16 nM. Eganelisib shows >100-fold selectivity over other lipid and protein kinases. | ||||||||||||||||||||
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Eganelisib (Standard) | ≥98% | Eganelisib (Standard) is the analytical standard of Eganelisib (HY-100716). This product is intended for research and analytical applications. Eganelisib (IPI549) is a potent and selective PI3Kγ inhibitor with an IC50 of 16 nM. Eganelisib shows >100-fold selectivity over other lipid and protein kinases. | ||||||||||||||||||||
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References
Keywords
