1808951-93-0
1808951-93-0
Chemical Structure
LP99
- CAS No.: 1808951-93-0
- Formula:C26H30ClN3O4S
- Molecular Weight:516.05
IUPAC Name: N-((2R,3S)-2-(4-chlorophenyl)-1-(1,4-dimethyl-2-oxo-1,2-dihydroquinolin-7-yl)-6-oxopiperidin-3-yl)-2-methylpropane-1-sulfonamide
InChIKey: LVDRREOUMKACNJ-BKMJKUGQSA-N
SMILES: O=C1N(C2=CC(N(C)C(C=C3C)=O)=C3C=C2)[C@H](C4=CC=C(Cl)C=C4)[C@@H](NS(CC(C)C)(=O)=O)CC1
Biological Activity: LP99, an epigenetic probe, is a potent and selective inhibitor of the BRD7 and BRD9 bromodomains with a Kd of 99 nM against BRD9. LP99 disrupts the binding of BRD7 and BRD9 to chromatin in cells[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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LP99 | 99.18% | LP99, an epigenetic probe, is a potent and selective inhibitor of the BRD7 and BRD9 bromodomains with a Kd of 99 nM against BRD9. LP99 disrupts the binding of BRD7 and BRD9 to chromatin in cells. | ||||||||||||||||||||
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References
Keywords
