182417-73-8
Chemical Structure
DPI-3290
Synonym(s): Org 41793
- CAS No.: 182417-73-8
- Formula:C30H34FN3O2
- Molecular Weight:487.61
IUPAC Name: 3-((R)-((2S,5R)-4-allyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)-N-(3-fluorophenyl)-N-methylbenzamide
InChIKey: LZXRQLIIMYJZDA-UETOGOEVSA-N
SMILES: O=C(N(C1=CC=CC(F)=C1)C)C2=CC=CC([C@@H](N3[C@@H](C)CN(CC=C)[C@H](C)C3)C4=CC=CC(O)=C4)=C2
Biological Activity: DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively. DPI-3290 is one of a series of novel centrally acting agents with potent antinociceptive activity[1].
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DPI-3290 | DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively. DPI-3290 is one of a series of novel centrally acting agents with potent antinociceptive activity. | |||||||||||||||||||||
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Keywords
