1. GPCR/G Protein
    Neuronal Signaling
  2. Opioid Receptor
  3. DPI-3290

DPI-3290 (Synonyms: Org 41793)

Cat. No.: HY-19231
Handling Instructions

DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively。DPI-3290 is one of a series of novel centrally acting agents with potent antinociceptive activity.

For research use only. We do not sell to patients.

DPI-3290 Chemical Structure

DPI-3290 Chemical Structure

CAS No. : 182417-73-8

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Description

DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively。DPI-3290 is one of a series of novel centrally acting agents with potent antinociceptive activity[1].

IC50 & Target

IC50: 0.18 nM (δ-opioid receptor), 0.46 nM (μ-opioid receptor) and 0.62 nM (κ-opioid receptor)[1]

In Vivo

DPI-3290 (Org 41793) (intravenous; 0.05 mg/kg) produces a 50% antinociceptive response in rats[1].

Molecular Weight

487.61

Formula

C₃₀H₃₄FN₃O₂

CAS No.

182417-73-8

SMILES

O=C(N(C1=CC=CC(F)=C1)C)C2=CC=CC([[email protected]@H](N3[[email protected]@H](C)CN(CC=C)[[email protected]](C)C3)C4=CC=CC(O)=C4)=C2

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Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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DPI-3290
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