2079886-19-2
2079886-19-2
Chemical Structure
GSK4028
- CAS No.: 2079886-19-2
- Formula:C17H21BrN4O
- Molecular Weight:377.28
IUPAC Name: 4-bromo-2-methyl-5-(((3S,5S)-1-methyl-5-phenylpiperidin-3-yl)amino)pyridazin-3(2H)-one
InChIKey: VZAFGXCWAWRULT-KGLIPLIRSA-N
SMILES: BrC1=C(N[C@H]2C[C@@H](C3=CC=CC=C3)CN(C)C2)C=NN(C)C1=O
Biological Activity: GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.
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GSK4028 | 98.06% | GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. | ||||||||||||||||||||
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GSK4028 (Standard) | ≥98% | GSK4028 (Standard) is the analytical standard of GSK4028 (HY-101027A). This product is intended for research and analytical applications. GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. | ||||||||||||||||||||
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Keywords
