2378173-15-8
2378173-15-8
Chemical Structure
PF-06928215
- CAS No.: 2378173-15-8
- Formula:C20H20N4O4
- Molecular Weight:380.40
IUPAC Name: (1R,2S)-2-(7-hydroxy-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamido)cyclohexane-1-carboxylic acid
InChIKey: PHGTYMRDHDEHLI-HIFRSBDPSA-N
SMILES: OC1=CC(C2=CC=CC=C2)=NC3=C(C(N[C@H]4CCCC[C@H]4C(O)=O)=O)C=NN13
Biological Activity: PF-06928215 is a cGAS (cyclic GMP-AMP Synthase) inhibitor with an IC50 of 4.9 μΜ. PF-06928215 has a high binding affinity of 0.2 μM (Kd)[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PF-06928215 | 99.68% | PF-06928215 is a cGAS (cyclic GMP-AMP Synthase) inhibitor with an IC50 of 4.9 μΜ. PF-06928215 has a high binding affinity of 0.2 μM (Kd). | ||||||||||||||||||||
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References
Keywords
