2408297-80-1

EP3 antagonist 4 Chemical Structure
2408297-80-1

Chemical Structure

EP3 antagonist 4

  • CAS No.: 2408297-80-1
  • Formula:C22H20Cl3FN4O3S2
  • Molecular Weight:577.91

IUPAC Name: (Z)-5-chloro-N-((2-(1-(2,4-dichlorobenzyl)-1,4,5,6-tetrahydro-7H-indazol-7-ylidene)-2-fluoroethyl)carbamoyl)-4-methylthiophene-2-sulfonamide

InChIKey: FYUOIRIANAUUOH-VLGSPTGOSA-N

SMILES: O=S(NC(NC/C(F)=C1CCCC(C=N2)=C\1N2CC3=C(C=C(C=C3)Cl)Cl)=O)(C4=CC(C)=C(S4)Cl)=O

Biological Activity: EP3 antagonist 4 (Compound 28) is an EP3 antagonist, with a Ki value of 2 nM for hEP. EP3 antagonist 4 shows low in vivo clearance, high oral AUC, and good bioavailability in the rat full PK studies. EP3 antagonist 4 can be used for research of beta cell dysfunction in diabetes[1].

Cat. No. Product Name Purity Description Pricing
HY-153256 		EP3 antagonist 4 EP3 antagonist 4 (Compound 28) is an EP3 antagonist, with a Ki value of 2 nM for hEP. EP3 antagonist 4 shows low in vivo clearance, high oral AUC, and good bioavailability in the rat full PK studies. EP3 antagonist 4 can be used for research of beta cell dysfunction in diabetes.
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