2682255-44-1
Chemical Structure
A031
- CAS No.: 2682255-44-1
- Formula:C50H61ClN10O7S
- Molecular Weight:981.60
IUPAC Name: 7-chloro-4H-benzo[e][1,2,4]thiadiazine 1,1-dioxide
InChIKey: PGVTULUCNZWYPD-YRHZNJHBSA-N
SMILES: O=C(N([C@@H]1C2)[C@H](CC1)C[C@@H]2OC3=CC(Cl)=C(C=C3)C#N)C4=CN=C(N5CCN(CC5)CCOCC(N[C@@H](C(C)(C)C)C(N6[C@@H](C[C@H](C6)O)C(N[C@H](C7=CC=C(C8=C(N=CS8)C)C=C7)C)=O)=O)=O)N=C4
Biological Activity: A031 is a PROTAC degrader targeting the androgen receptor. A031 induces time-dependent degradation of androgen receptor protein. A031 exerts tumor growth inhibitory effects in a zebrafish model xenografted with human prostate cancer cells. A031 can be used in studies related to prostate cancer[1].
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A031 | A031 is a PROTAC degrader targeting the androgen receptor. A031 induces time-dependent degradation of androgen receptor protein. A031 exerts tumor growth inhibitory effects in a zebrafish model xenografted with human prostate cancer cells. A031 can be used in studies related to prostate cancer. | |||||||||||||||||||||
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Keywords
