2747914-87-8
2747914-87-8
Chemical Structure
N-Desmethyl Azelastine-d4-1
- CAS No.: 2747914-87-8
- Formula:C21H18D4ClN3O
- Molecular Weight:371.90
IUPAC Name: 4-(methyl-d3)benzaldehyde-2,3,5,6-d4
InChIKey: WRYCMIFVXDQIKN-NMRLXUNGSA-N
SMILES: O=C1N(C2CCNCCC2)N=C(CC3=CC=C(Cl)C=C3)C4=C1C([2H])=C([2H])C([2H])=C4[2H]
Biological Activity: N-Desmethyl Azelastine-d4-1 is the deuterium labeled N-Desmethyl Azelastine[1].
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N-Desmethyl Azelastine-d4-1 | N-Desmethyl Azelastine-d4-1 is the deuterium labeled N-Desmethyl Azelastine. | |||||||||||||||||||||
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Desmethylazelastine | Desmethylazelastine is a main active metabolite of Azelastine that is oxidatively metabolized by the cytochrome P450 enzyme system with a protein binding rate of 97% and an elimination half-life of 54 hours. Azelastine is an orally active, selective and high-affinity histamine H1-receptor antagonist. Azelastine can be used in studies of allergic rhinitis, asthma, diabetic hyperlipidemic and SARS-CoV-2. | |||||||||||||||||||||
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References
