2924415-92-7
2924415-92-7
Chemical Structure
Ack1 inhibitor 1
- CAS No.: 2924415-92-7
- Formula:C39H40F3N7O4
- Molecular Weight:727.77
InChIKey: RONKBVWJPIOCJX-WJOKGBTCSA-N
SMILES: CN(CC1)CCN1C(C=C2)=CC(OCC)=C2NC3=NC=C4C(N(C[C@@H]5OCCC5)C(C(C6=CC(NC(C7=CC(C(F)(F)F)=CC=C7)=O)=CC=C6)=C4)=O)=N3
Biological Activity: Ack1 inhibitor 1 is a potent, selective, and orally active inhibitor of ACK1 kinase with an IC50 value of 2.1 nM. Ack1 inhibitor 1 inhibits the phosphorylation of ACK1 and activation of downstream AKT. Ack1 inhibitor 1 has anti-tumor activity[1].
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Ack1 inhibitor 1 | Ack1 inhibitor 1 is a potent, selective, and orally active inhibitor of ACK1 kinase with an IC50 value of 2.1 nM. Ack1 inhibitor 1 inhibits the phosphorylation of ACK1 and activation of downstream AKT. Ack1 inhibitor 1 has anti-tumor activity. | |||||||||||||||||||||
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References
Keywords
