3032642-29-5
3032642-29-5
Chemical Structure
EGFR/ACK1-IN-1
- CAS No.: 3032642-29-5
- Formula:C22H20ClN7O
- Molecular Weight:433.89
InChIKey: FCHNDUSRWAGJES-UHFFFAOYSA-N
SMILES: ClC1=CC=C(C2=C1)N=C(N=C2NC3=CC=CC(NC(C=C)=O)=C3)NC4=CN(N=C4)CC
Biological Activity: EGFR T790M/L858R/ACK1-IN-1 is a dual inhibitor of EGFR T790M/L858R and ACK1. IC50 values are 23 and 263 nM, respectively. EGFR T790M/L858R/ACK1-IN-1 can inhibit cell proliferation and has antitumor activity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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EGFR/ACK1-IN-1 | 98.19% | EGFR T790M/L858R/ACK1-IN-1 is a dual inhibitor of EGFR T790M/L858R and ACK1. IC50 values are 23 and 263 nM, respectively. EGFR T790M/L858R/ACK1-IN-1 can inhibit cell proliferation and has antitumor activity. | ||||||||||||||||||||
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References
Keywords
