3054869-10-9
3054869-10-9
Chemical Structure
PI3Kδ/BET-IN-1
- CAS No.: 3054869-10-9
- Formula:C27H34N6O3S
- Molecular Weight:522.66
SMILES: CN1C=C(C2=NC(N3CCOCC3)=C4SC(CN5CCC(C(C)(O)C)CC5)=CC4=N2)C6=C(C1=O)NC=C6
Biological Activity: PI3Kδ/BET-IN-1 (compound 10b) shows excellent and balanced activities against PI3Kδ (IC50 = 112 nM) and BRD4-BD1 (IC50 = 19 nM) and exhibits strong antiproliferative activities in DLBCL cells[1].
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PI3Kδ/BET-IN-1 | PI3Kδ/BET-IN-1 (compound 10b) shows excellent and balanced activities against PI3Kδ (IC50 = 112 nM) and BRD4-BD1 (IC50 = 19 nM) and exhibits strong antiproliferative activities in DLBCL cells. | |||||||||||||||||||||
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References
Keywords
