319492-82-5
319492-82-5
Chemical Structure
GAK inhibitor 49
- CAS No.: 319492-82-5
- Formula:C20H22N2O5
- Molecular Weight:370.40
IUPAC Name: 6,7-dimethoxy-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine
InChIKey: VYPGLYMWNDRFGZ-UHFFFAOYSA-N
SMILES: COC1=C(OC)C(OC)=CC(NC2=CC=NC3=CC(OC)=C(OC)C=C23)=C1
Biological Activity: GAK inhibitor 49 is a potent, ATP-competitive and highly selective cyclin G associated kinase (GAK) inhibitor with a Ki of 0.54 nM and a cell IC50 of 56 nM. GAK inhibitor 49 also shows binding to RIPK2[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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GAK inhibitor 49 | 98.28% | GAK inhibitor 49 is a potent, ATP-competitive and highly selective cyclin G associated kinase (GAK) inhibitor with a Ki of 0.54 nM and a cell IC50 of 56 nM. GAK inhibitor 49 also shows binding to RIPK2. | ||||||||||||||||||||
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References
Keywords
