408305-09-9
408305-09-9
Chemical Structure
Ac-RYYRWK-NH2 TFA
- CAS No.: 408305-09-9
- Formula:C51H70F3N15O11
- Molecular Weight:1126.19
InChIKey: VNWKTOKETHGBQD-UHFFFAOYSA-N
SMILES: OC(C(F)(F)F)=O.OC(C=C1)=CC=C1C[C@H](NC([C@@H](NC([C@@H](NC(C)=O)CCCNC(N)=N)=O)CC2=CC=C(C=C2)O)=O)C(N[C@@H](CCCNC(N)=N)C(N[C@H](C(N[C@H](C(N)=O)CCCCN)=O)CC3=CNC4=CC=CC=C34)=O)=O
Biological Activity: Ac-RYYRWK-NH2 is a potent and selective partial agonist for the nociceptin receptor (NOP), [3H]Ac-RYYRWK-NH2 binds to rat cortical membranes ORL1 with a Kd of 0.071 nM, but has no affinity for μ-, κ- or δ-opioid receptors[1].
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Ac-RYYRWK-NH2 TFA | Ac-RYYRWK-NH2 is a potent and selective partial agonist for the nociceptin receptor (NOP), [3H]Ac-RYYRWK-NH2 binds to rat cortical membranes ORL1 with a Kd of 0.071 nM, but has no affinity for μ-, κ- or δ-opioid receptors. | |||||||||||||||||||||
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References
Keywords
