1. GPCR/G Protein
    Neuronal Signaling
  2. Opioid Receptor
  3. Ac-RYYRWK-NH2 TFA

Ac-RYYRWK-NH2 TFA 

Cat. No.: HY-P1316A
Handling Instructions

Ac-RYYRWK-NH2 is a potent and selective partial agonist for the nociceptin receptor (NOP), [3H]Ac-RYYRWK-NH2 binds to rat cortical membranes ORL1 with a Kd of 0.071 nM, but has no affinity for µ-, κ- or δ-opioid receptors.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

Ac-RYYRWK-NH2 TFA Chemical Structure

Ac-RYYRWK-NH2 TFA Chemical Structure

CAS No. : 408305-09-9

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Description

Ac-RYYRWK-NH2 is a potent and selective partial agonist for the nociceptin receptor (NOP), [3H]Ac-RYYRWK-NH2 binds to rat cortical membranes ORL1 with a Kd of 0.071 nM, but has no affinity for µ-, κ- or δ-opioid receptors[1].

In Vitro

[3H]ac-RYYRWK-NH2 binding to rat cortical membranes revealed a single high affinity site for [3H]ac-RYYRWK-NH2 (Kd=0.071 nM)[1].
Naloxone benzoylhydrazone displaced [3H]acRYYRWK-NH2 binding to rat cortical membranes (Ki=104 nM) and human ORL1 (Ki=136 nM) as well as [125I]Tyr14-NC-OH to ORL1 (Ki=37 nM) has no affinity for µ-, κ- or δ-opioid receptors[1].

Molecular Weight

1126.19

Formula

C₅₁H₇₀F₃N₁₅O₁₁

CAS No.

408305-09-9

Sequence Shortening

Ac-RYYRWK-NH2

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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

Ac-RYYRWK-NH2Opioid ReceptorInhibitorinhibitorinhibit

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Ac-RYYRWK-NH2 TFA
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