850665-21-3
850665-21-3
Chemical Structure
GSK248233A
- CAS No.: 850665-21-3
- Formula:C25H24N8O3
- Molecular Weight:484.51
InChIKey: KODFUVBIVXFWPF-UHFFFAOYSA-N
SMILES: O=C(C1=CC=C(N(C)C)C=C1)NC2=CC(OC3=CC(N(CC)C(C4=NON=C4N)=N5)=C5C=N3)=CC=C2
Biological Activity: GSK248233A is a dual inhibitor of Fluc and VEGFR2 with IC50 of 1.03 μM and 2 nM, respectively. GSK248233A also shows activity against the AGC family. GSK248233A acts as a protein kinase inhibitor across ATP-dependent and -independent luciferases with potential implications for Fluc reporter assays[1].
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GSK248233A | GSK248233A is a dual inhibitor of Fluc and VEGFR2 with IC50 of 1.03 μM and 2 nM, respectively. GSK248233A also shows activity against the AGC family. GSK248233A acts as a protein kinase inhibitor across ATP-dependent and -independent luciferases with potential implications for Fluc reporter assays. | |||||||||||||||||||||
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References
Keywords
